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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10694 | CB1 inverse agonist 1 | MRL-650 | Cannabinoid Receptor |
CB1 inverse agonist 1 (MRL-650) is an orally active and selective CB1 agonist. The IC50s for CB1 and CB2 are 7.5 nM and 4100 nM, respectively. CB1 inverse agonist 1 shows anorexigenic effects. | |||
T13080L | Taranabant | MK-0364 | Cannabinoid Receptor |
Taranabant (MK-0364) is a selective and potent cannabinoid 1 (CB1) receptor inverse agonist used in the study of obesity and nicotine dependence. | |||
T1519L | Rimonabant | SR141716 | Cannabinoid Receptor , Antibacterial , Acyltransferase |
Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1. It is an anorectic anti-obesity drug produced and marketed by Sanofi-Aventis. Its main avenue of effect is a reduction in appetite. Rimonabant... | |||
T13081 | Taranabant racemate | MK-0364 racemate | Cannabinoid Receptor |
Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor. | |||
T62180 | CB1/2 agonist 2 | ||
CB1/2 agonist 2 (compound 23) is a potent non-selective cannabinoid ligand with Ki of 3.5 nM and 1.2 nM, respectively. CB1/2 agonist 2 is a full agonist of CB1 and a competitive inverse agonist of CB2. BACE-IN-1 is a com... | |||
T75799 | Hemopressin(human, mouse) TFA | Cannabinoid Receptor | |
Hemopressin TFA, a nonapeptide originating from the α1-chain of hemoglobin and initially isolated from rat brain homogenates, is an orally active, selective inverse agonist of CB1 cannabinoid receptors that demonstrates ... | |||
T75798 | Hemopressin(rat) TFA | ||
Hemopressin(rat) TFA, a nonapeptide originating from the α1-chain of hemoglobin, was first isolated from rat brain homogenates. It acts as an orally active, selective, and inverse agonist of the CB1 cannabinoid receptors... |